Research areas

  1. Published

    High resolution crystal structures of the p120 RasGAP SH3 domain

    Ross, B., Kristensen, O., Favre, D., Walicki, J., Kastrup, Jette Sandholm Jensen, Widmann, C. & Gajhede, Michael, 2007, In: Biochemical and Biophysical Research Communications. 353, 2, p. 463-468

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Structural and functional studies in allergy and signal transduction

    Ross, B., 2007, København: Det Farmaceutiske Fakultet. 134 p.

    Research output: Book/ReportPh.D. thesisResearch

  3. Published

    Nanoporous magnesium aluminometasilicate tablets for precise, controlled, and continuous dosing of chemical reagents and catalysts: applications in parallel solution-phase synthesis

    Ruhland, T., Nielsen, S. D., Holm, P. & Christensen, C. H., 2007, In: Journal of Combinatorial Chemistry. 9, 2, p. 301-305

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Multi-component and multi-class analysis of 23 antimicrobials, metabolites and degradation products

    Runnqvist, H. E. S., Krogh, K. A., Halling-Sørensen, B. & Jensen, L. B., 2007.

    Research output: Contribution to conferencePosterResearch

  5. Published

    Teaching social sciences to undergraduate pharmacy students: An international survey

    Ryan, K., Bissell, P., Anderson, C., Traulsen, Janine Marie & Sleath, B., 2007, In: Pharmacy Education. 1, p. 1-9

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Dynamics of water molecules in the active-site cavity of human cytochromes P450

    Rydberg, P., Rod, T. H., Olsen, L. & Ryde, U., 2007, In: Journal of Physical Chemistry Part B: Condensed Matter, Materials, Surfaces, Interfaces & Biophysical. 111, 19, p. 5445-5457

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    General transition-state force field for cytochrome P450 hydroxylation

    Rydberg, P. Å. A., Olsen, L., Norrby, P. & Ryde, U., 2007, In: Journal of Chemical Theory and Computation. 3, 5, p. 1765-1773

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Solid-state transformation of erythromycin A dihydrate during drying monitored by near infared spectroscopy

    Römer, M., Heinämäki, J., Miroshnyk, I., Kivikero, N., Sandler, N., Rantanen, Jukka & Yliruusi, J., 2007, In: European Journal of Pharmaceutical Sciences. 32S, 1, p. S48

    Research output: Contribution to journalConference abstract in journalResearch

  9. Published

    Phase transformations of erythromycin A dihydrate during pelletisation and drying

    Römer, M., Heinämäki, J., Miroshnyk, I., Sandler, N., Rantanen, Jukka & Yliruusi, J., 2007, In: European Journal of Pharmaceutics and Biopharmaceutics. 67, 1, p. 246-252

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Biodegradation of selected emerging organic contaminants in the environment: an overview

    Sarmah, A. K. & Halling-Sørensen, B., 2007, Leading-edge environmental biodegradation. Pawley, L. E. (ed.). Nova Science Publishers, p. 53-93

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  11. Published

    Probing insulin's secondary structure after entrapment into alginate/chitosan nanoparticles

    Sarmento, B., Ferreira, D. C., Jørgensen, Lene & van de Weert, Marco, 2007, In: European Journal of Pharmaceutics and Biopharmaceutics. 65, 1, p. 10-17

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Determination of amorphous content in the pharmaceutical process environment

    Savolainen, M., Jouppila, K., Pajamo, O., Christiansen, L., Strachan, C., Karjalainen, M. & Rantanen, Jukka, 2007, In: Journal of Pharmacy and Pharmacology. 59, 2, p. 161-170

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    Energy substrates to support glutamatergic and GABAergic synaptic function: Role of glycogen, glucose and lactate

    Schousboe, Arne, Bak, Lasse Kristoffer, Sickmann, H. M., Sonnewald, U. & Waagepetersen, Helle S., 2007, In: Neurotoxicity Research. 12, 4, p. 263-268

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. Published

    GABA: Homeostatic and pharmacological aspects

    Schousboe, Arne & Waagepetersen, Helle S., 2007, In: Progress in Brain Research. 160, p. 9-19

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    Calcimimetic, AMG 073, induces relaxtion on isolated rat aorta

    Smajilovic, S., Sheykhzade, Majid, Holmegard, H. N., Haunso, S. & Tfelt-Hansen, J., 2007, In: Vascular Pharmacology. 47, p. 222-228

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Multivariate toxicity screening of liposomal formulations on a human buccal cell line

    Smidstad, G., Jacobsen, Jette & Sande, S. A., 2007, In: Internation Journal of Pharmaceutics. 330, 1-2, p. 14-22

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    Actions of toxins on cerebral metabolism at cellular level

    Sonnewald, U., Syversen, T., Schousboe, Arne, Waagepetersen, Helle S. & Aschner, M., 2007, Handbook of Neurochemistry and Molecular Neurobiology: Brain Energetics. Integration of Molecular and Cellular Processes. Lajtha, A., Gibson, G. E. & Dienel, G. A. (eds.). 3rd. ed. ed. Berlin: Springer, Vol. 3. p. 569-585

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  18. Published

    Determination of abiotic and microbial transformation products of ivermectin

    Sporring, S. H., Krogh, K. A., Jensen, G. G., Raich-Montiu, J. & Halling-Sørensen, B., 2007.

    Research output: Contribution to conferencePosterResearch

  19. Published

    Targeted natural product isolation guided by HPLC-SPE-NMR: constituents of Hubertia species

    Sprogøe, K., Stærk, Dan, Jäger, A. K., Adsersen, A., Hansen, S. H., Witt, M., Landbo, A. R., Meyer, A. S. & Jaroszewski, J. W., 2007, In: Journal of Natural Products. 70, 9, p. 1472-1477

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    Differential effect of opioids in patients with chronic pancreatitis: an experimental pain study

    Staahl, C., Dimcevski, G., Andersen, S. D., Thorsgaard, N., Christrup, Lona Louring, Arendt-Nielsen, L. & Drewes, A. M., 2007, In: Scandinavian Journal of Gastroenterology. 42, 3, p. 383-90

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Monoamine oxidase inhibition by southern african traditional medicinal plants

    Stafford, G. I., Pedersen, P. D., Jäger, A. K. & van Staden, J., 2007, In: South African Journal of Botany. 73, 3, p. 384-390

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Lægemiddelformen og formuleringens indflydelse på den terapeutiske effekt af lægemidler

    Steffansen, B., 2007, In: Lægemiddelkataloget. p. 39-45

    Research output: Contribution to journalJournal articleCommissioned

  23. Published

    Characterisation and physical stability of PEGylated glucagon

    Stigsnæs, P., Frøkjær, Sven, Bjerregaard, S., van de Weert, Marco, Kingshott, P. & Møller, E. H., 2007, In: Internation Journal of Pharmaceutics. 330, 1-2, p. 89-98

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Insight into the metastable form of theophylline monohydrate using vibrational spectroscopy, computational chemistry and multivariate analysis

    Strachan, C. J., Howell, S. L., Aaltonen, J., Heinz, A., Kogermann, K. & Rantanen, Jukka, 2007, In: European Journal of Pharmaceutical Sciences. 32, 1, p. S8

    Research output: Contribution to journalConference abstract in journalResearch

  25. Published

    Raman spectroscopy for quantitative analysis of pharmaceutical solids

    Strachan, C. J., Rades, Thomas, Gordon, K. C. & Rantanen, Jukka, 2007, In: Journal of Pharmacy and Pharmacology. 59, 2, p. 179-192

    Research output: Contribution to journalJournal articleResearchpeer-review

  26. Published

    A pilot study of pharmacist-initiated interventions in drug therapy in an Australian paediatric hospital

    Struck, P., Pedersen, K. H., Moodley, P. & Rasmussen, M., 2007, In: EJHP Science. 13, 4, p. 105-112

    Research output: Contribution to journalJournal articleResearchpeer-review

  27. Published

    Noter til M25-1 spektroskopi

    Stærk, Dan & Jaroszewski, J. W., 2007, København: Københavns Universitet, Det Farmaceutiske Fakultet, Institut for Medicinalkemi. 49 p.

    Research output: Book/ReportCompendium/lecture notesEducation

  28. Published

    Selektive lægemiddelstoffer designet ud fra krystalstrukturer

    Szymanska, E. M. & Johansen, Tommy Nørskov, 2007, In: Lægemiddelforskning. p. 34-35

    Research output: Contribution to journalJournal articleCommunication

  29. Published

    Risk assessment of topically applied products

    Søborg, T., Basse, L. H. & Halling-Sørensen, B., 2007, In: Toxicology. 236, 1-2, p. 140-148

    Research output: Contribution to journalJournal articleResearchpeer-review

  30. Published

    I-125 used for labelling of proteins in an absorption model changes the absorption rate of insulin aspart

    Søhoel, A., Plum, A., Frøkjær, Sven & Thygesen, P., 2007, In: Internation Journal of Pharmaceutics. 330, 1-2, p. 114-120

    Research output: Contribution to journalJournal articleResearchpeer-review

  31. Published

    Structures of OppA and PstS from Yersinia pestis indicate variability of interactions with transmembrane domains

    Tanabe, M., Mirza, Osman Asghar, Bertrand, T., Atkins, H. S., Titball, R. W., Iwata, S., Brown, K. A. & Byrne, B., 2007, In: Acta Crystallographica. Section D: Biological Crystallography. 63, 11, p. 1185-1193

    Research output: Contribution to journalJournal articleResearchpeer-review

  32. Published

    Kan danske registre anvendes ved utilsigtede haendelser ved type 2-diabetes?

    Thomsen, L. A., Gundgaard, J., Søndergaard, B., Melander, A. & Sørensen, J., 2007, In: Ugeskrift for læger. 169, 33, p. 2637-42

    Research output: Contribution to journalJournal articleResearchpeer-review

  33. Published

    Systematic review of the incidence and characteristics of preventable adverse drug events in ambulatory care

    Thomsen, L. A., Winterstein, A. G., Søndergaard, B., Nørgaard, Lotte Stig & Melander, A., 2007, In: Annals of Pharmacotherapy. 41, 9, p. 1411-26

    Research output: Contribution to journalJournal articleResearchpeer-review

  34. Published

    Involvement of Y5 receptors in neuropeptide Y agonist-induced analgesic-like effect in the rat hot plate test

    Thomsen, M., Wörtwein, Gitta, Olesen, M. V., Begtrup, M., Havez, S., Bolwig, T. G. & Woldbye, David Paul Drucker, 2007, In: Brain Research. 1155, p. 49-55

    Research output: Contribution to journalJournal articleResearchpeer-review

  35. Published

    Design, synthesis, and evaluation of tripeptidic promoieties targeting the intestinal peptide transporter hPEPT1

    Thorn, K., Andersen, R., Christensen, J., Jacobsen, P., Nielsen, C. U., Steffansen, B. & Begtrup, M., 2007, In: ChemMedChem. 2, 4, p. 479-487

    Research output: Contribution to journalJournal articleResearchpeer-review

  36. Published

    Transportpeptider: nøglen til forbedret optagelse af lægemiddelstoffer

    Thorn, K., Nielsen, C. U. & Begtrup, M., 2007, In: Lægemiddelforskning. p. 18-19

    Research output: Contribution to journalJournal articleCommunication

  37. Published

    Characterization and physical stability of tolfenamic acid-PVP K30 solid dispersions

    Thybo, P., Kristensen, J. & Hovgaard, L., 2007, In: Pharmaceutical Development and Technology. 12, 1, p. 43-53

    Research output: Contribution to journalJournal articleResearchpeer-review

  38. Published

    Antioxidant activity of cichoric acid and alkamides from Echinacea purpurea, alone and in combination

    Thygesen, L., Thulin, J., Mortensen, A., Skibsted, Leif Horsfelt & Mølgaard, Per, 2007, In: Food Chemistry. 101, 1, p. 74-81 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  39. Published

    Influence of polymorphic form, morphology, and excipient interactions on the dissolution of carbamazepine compacts

    Tian, F., Sandler, N., Aaltonen, J., Lang, C., Saville, D. J., Gordon, K. C., Strachan, C. J., Rantanen, Jukka & Rades, Thomas, 2007, In: Journal of Pharmaceutical Sciences. 96, 3, p. 584-594

    Research output: Contribution to journalJournal articleResearchpeer-review

  40. Published

    Antiplasmodial and prehemolytic activities of alpha-peptide-beta-peptoid chimeras

    Vedel, L., Bonke, G., Foged, Camilla, Ziegler, H. L., Franzyk, Henrik, Jaroszewski, J. W. & Olsen, Christian Adam, 2007, In: ChemBioChem. 8, 15, p. 1781-1784 4 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  41. Published

    A helical structural nucleus is the primary elongating unit of insulin amyloid fibrils

    Vestergaard, Bente, Jensen, M. G., Roessle, M., Kastrup, Jette Sandholm Jensen, van de Weert, Marco, Flink, J. M., Frøkjær, Sven, Gajhede, Michael & Svergun, D. I., 2007, In: PLoS - Biology. 5, 5, p. 1089-1097

    Research output: Contribution to journalJournal articleResearchpeer-review

  42. Published

    Differences in kinetics of structurally related competitive GABAA receptor antagonists

    Vestergaard, H. T., Cannillo, C., Frølund, Bente & Kristiansen, Uffe, 2007, In: Neuropharmacology. 52, 3, p. 873-882

    Research output: Contribution to journalJournal articleResearchpeer-review

  43. Published

    Pharmacokinetics of morphine-6-glucuronide following oral administration in healthy volunteers

    Villesen, H. H., Kristensen, K., Hansen, S. H., Jensen, N., Skram, U. & Christrup, Lona Louring, 2007, In: European Journal of Clinical Pharmacology. 63, 8, p. 761-767

    Research output: Contribution to journalJournal articleResearchpeer-review

  44. Published

    Pharmakonetics of morphine and oxycodone following intravenous administration in elderly patients

    Villesen, H. H., Banning, A., Petersen, R. H., Weinelt, S., Poulsen, J. B., Hansen, S. H. & Christrup, Lona Louring, 2007, In: Therapeutics and Clinical Risk Management. 3, 5

    Research output: Contribution to journalJournal articleResearchpeer-review

  45. Published

    A tetrazolyl-substituted subtype-selective AMPA receptor agonist

    Vogensen, S. B., Frydenvang, Karla Andrea, Greenwood, J. R., Postorino, G., Nielsen, Birgitte, Pickering, Darryl S, Ebert, B., Bølcho, U., Egebjerg, J., Gajhede, Michael, Kastrup, Jette Sandholm Jensen, Johansen, Tommy Nørskov, Clausen, Rasmus Prætorius & Krogsgaard-Larsen, Povl, 2007, In: Journal of Medicinal Chemistry. 50, 10, p. 2408-2414

    Research output: Contribution to journalJournal articleResearchpeer-review

  46. Published

    Glutamine, glutamate and GABA: metabolic aspects

    Waagepetersen, Helle S., Sonnerwald, U. & Schousboe, Arne, 2007, Handbook of neurochemistry and molecular neurobiology: amino acids and peptides in the nervous system. Lajtha, A., Oja, S. S., Schousboe, A. & Saransaari, P. (eds.). 3rd. ed. Berlin: Springer, p. 1-21

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  47. Published

    One third of glycolytic activity in astrocytes depends on the operation of the glycogen shunt

    Walls, Anne Byriel, Heimbürger, C. M., Sickmann, H. M., Bouman, S. D., Schousboe, Arne & Waagepetersen, Helle S., 2007, In: Journal of Neurochemistry. 102, s1, p. 119

    Research output: Contribution to journalConference abstract in journalResearch

  48. Published

    Effects of spinal cord stimulation on peripheral blood circulation in rats with streptozotocin-induced diabetes

    Wu, M., Ghorbani, M. L. M., Qin, C., Farber, J. P., Linderoth, B. & Foreman, R. D., 2007, In: Neuromodulation: Technology at the Neural Interface. 10, 3

    Research output: Contribution to journalJournal articleResearchpeer-review

  49. Published

    Characterisation of salmon calcitonin in spray-dried powder for inhalation. Effect of chitosan

    Yang, Mingshi, Velaga, S., Yamamoto, H., Takeuchi, H., Kawashima, Y., Hovgaard, L., van de Weert, Marco & Frøkjær, Sven, 2007, In: Internation Journal of Pharmaceutics. 331, 2, p. 176-181

    Research output: Contribution to journalJournal articleResearchpeer-review

  50. Published

    Activation of ERK, JNK, Akt, and G-protein coupled signaling by hybrid angiotensin II AT1/bradykinin B2 receptors expressed in HEK-293 cells

    Yu, J., Lubinsky, D., Tsomaia, N., Huang, Z., Taylor, L., Mierke, D., Navarro, J., Mirza, Osman Asghar & Polgar, P., 2007, In: Journal of Cellular Biochemistry. 101, 1, p. 192-204

    Research output: Contribution to journalJournal articleResearchpeer-review

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