Research areas

  1. Published

    Ligands for the GABA recognition site at the GABAA receptor: Structure-activity studies

    Frølund, Bente, Kristiansen, Uffe, Krogsgaard-Larsen, Povl & Liljefors, T., 2008, Chemistry and molecular aspects of drug design and action. Rekka, E. A. & Kourounakis, P. N. (eds.). Boca Raton, Fl: CRC Press, p. 139-147

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  2. Published

    Lipid-based formulations for danazol containing a digestible surfactant, labrafil M2125CS: In vivo bioavailability and dynamic in vitro lipolysis

    Larsen, A., Holm, R., Pedersen, M. L. & Mullertz, Anette , 2008, In: Pharmaceutical Research. 25, 12, p. 2769-2777

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Liposome-mediated triggering of complement cascade

    Moghimi, S. M. & Hamad, I., 2008, In: Journal of Liposome Research. 18, 3, p. 195-209

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Lymphatic tageting of immuno-PEG-liposomes: Evaluation of antibody-coupling procedures on lymph node macrophage uptake

    Moghimi, S. M. & Moghimi, M., 2008, In: Journal of Drug Targeting. 16, 7-8, p. 586-590

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Lægemidler fra naturstoffer: fortid eller fremtid?

    Jaroszewski, J. W., Christensen, Søren Brøgger, Franzyk, Henrik, Stærk, Dan & Ziegler, H., 2008, In: Lægemiddelforskning. p. 4-6

    Research output: Contribution to journalJournal articleCommunication

  6. Published

    Lægemidlers effekt på fedtnedbrydning kan måles i rotter

    Mølhøj, S., Malmlöf, K., Johansen, T. & Hansen, Harald S., 2008, In: Lægemiddelforskning. p. 55-57

    Research output: Contribution to journalJournal articleCommunication

  7. Published

    MAO-A inhibitory activity of quercetin from Calluna vulgaris Hull

    Saaby, Lasse, Jäger, A. K. & Rasmussen, H. B., 2008.

    Research output: Contribution to conferencePosterResearch

  8. Published

    Metabolic activation of carboxylic acids

    Skonberg, C., Olsen, J., Madsen, K. G., Hansen, S. H. & Grillo, M. P., 2008, In: Expert Opinion on Drug Metabolism & Toxicology. 4, 4, p. 425-438

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Metabolic cleavage and translocation efficiency of selected cell penetrating peptides: A comparative study with epithelial cell cultures

    Foerg, C., Weller, K. M., Rechsteiner, H., Nielsen, Hanne Mørck, Fernandez-Carneado, J., Brunisholz, R., Giralt, E. & Merkle, H. P., 2008, In: The AAPS Journal. 10, 2, p. 349-359

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Metabolism of [1,6-13C]glucose and [U-13C]glutamine and depolarization induced GABA release in superfused mouse cerebral cortical mini-slices

    Waagepetersen, Helle S., Døring, S. & Schousboe, Arne, 2008, In: Neurochemical Research. 33, 8, p. 1610-1617

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Metabolism of [U-13C]glutamine and [U-13C]glutamate in isolated rat brain mitochondria suggests functional phosphate-activated glutaminase activity in matrix

    Bak, Lasse Kristoffer, Zieminska, E., Waagepetersen, Helle S., Schousboe, Arne & Albrecht, J., 2008, In: Neurochemical Research. 33, 2, p. 273-278

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Metode til screening af modificerede proteinlægemidler under opbevaring

    Petersen, C., Jørgensen, Lene, Hostrup, S., Bukrinsky, J. T. & Frøkjær, Sven, 2008, In: Lægemiddelforskning. p. 16-18

    Research output: Contribution to journalJournal articleCommunication

  13. Published

    Mild psychoactive constituents of Mentha aquatica L.

    Stafford, G. I., Almqvist, J. P., Vangsøe, S. A. K., Olsen, H. T., Christensen, Søren Brøgger, Adsersen, A., Jäger, A. K. & van Staden, J., 2008, In: South African Journal of Botany. 2, p. 389

    Research output: Contribution to journalConference abstract in journalResearch

  14. Published

    Modified peptides as potent inhibitors of the postsynaptic density-95/N-methyl-D-aspartate receptor interaction

    Bach, Anders, Chi, C. N., Olsen, T. B., Pedersen, S. W., Røder, M. U., Pang, G. F., Clausen, Rasmus Prætorius, Jemth, P. & Strømgaard, Kristian, 2008, In: Journal of Medicinal Chemistry. 51, 20, p. 6450-6459

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    Molecular interactions in lipophilic environments studied by electrochemistry at interfaces between immiscible electrolyte solutions

    Deryabina, M., Hansen, S. H. & Jensen, H., 2008, In: Analytical Chemistry. 80, 1, p. 203-208

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Molecular mechanism of agonist recognition by the ligand-binding core of the ionotropic glutamate receptor 4

    Kasper, C., Frydenvang, Karla Andrea, Naur, P., Gajhede, Michael, Pickering, Darryl S & Kastrup, Jette Sandholm Jensen, 2008, In: FEBS Letters. 582, 29, p. 4089-4094

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    N-Hydroxypyrazolyl glycine derivatives as selective N-methyl-D-aspartic acid receptor ligands

    Clausen, Rasmus Prætorius, Christensen, C., Hansen, K. B., Greenwood, J. R., Jørgensen, L., Micale, N., Madsen, J. C., Nielsen, Birgitte, Egebjerg, J., Bräuner, Hans, Traynelis, S. F. & Kristensen, Jesper Langgaard, 2008, In: Journal of Medicinal Chemistry. 51, 14, p. 4179-87

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    Near-infrared spectroscopy for cocrystal screening: a comparative study with Raman spectroscopy

    Allesø, M., Velaga, S., Alhalaweh, A., Cornett, Claus, Rasmussen, Morten Arendt, van der Berg, Franciscus Winfried J, de Diego, H. L. & Rantanen, Jukka, 2008, In: Analytical Chemistry. 80, 20, p. 7755-7764 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    Nedfrysning af immunceller kan overflødiggøre forsøgskaniner i lægemiddelkontrol

    Timm, M., Moesby, L. & Hansen, E. W., 2008, In: Lægemiddelforskning. p. 43-45

    Research output: Contribution to journalJournal articleCommunication

  20. Published

    New initiative for thematic issues: An invitation: Brief overview of the five "hot" themes in Ecological Modelliong

    Jørgensen, S. E., Grant, W. E., Legovic, T. & Nielsen, S. N., 2008, In: Ecological Modelling. p. 273-275

    Research output: Contribution to journalComment/debateResearch

  21. Published

    Novel acetylcholine and carbamoylcholine analogues: Development of a functionally selective a4ß2 nicotinic acetylcholine receptor agonist

    Hansen, C. P., Jensen, Anders A., Christensen, J. K., Balle, T., Liljefors, T. & Frølund, Bente, 2008, In: Journal of Medicinal Chemistry. 51, 23, p. 7380-7395

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Novel high-affinity and selective biaromatic 4-substituted ¿-hydroxybutyric acid (GHB) analogues as GHB ligands: design, synthesis, and binding studies

    Høg, S., Wellendorph, Petrine, Nielsen, Birgitte, Frydenvang, Karla Andrea, Dahl, I. F., Bräuner, Hans, Brehm, L., Frølund, Bente & Clausen, Rasmus Prætorius, 2008, In: Journal of Medicinal Chemistry. 51, 24, p. 8088-8095

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    Novel wound models for characterizing ibuprofen release from foam dressings

    Steffansen, B. & Herping, S. P. K., 2008, In: Internation Journal of Pharmaceutics. 364, 1, p. 150-155

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Ny human GABA-transportør: et muligt mål for behandling af epilepsi

    Christiansen, B., Kvist, T., Jensen, Anders A. & Bräuner, Hans, 2008, In: Lægemiddelforskning. p. 25-27

    Research output: Contribution to journalJournal articleCommunication

  25. Published

    Nye depotlægemidler til injektion i gigtramte led: kan laboratoriemodeller reducere antallet af dyreforsøg

    Frost, A. B., Larsen, Susan Weng, Østergaard, Jesper & Larsen, C. S., 2008, In: Lægemiddelforskning. p. 46-48

    Research output: Contribution to journalJournal articleCommunication

  26. Published

    On the mechanism of drug release from oil suspensions in vitro using local anasthetics as model drug compounds

    Larsen, Susan Weng, Frost, A. B., Østergaard, Jesper, Marcher, H. & Larsen, C. S., 2008, In: European Journal of Pharmaceutical Sciences. 34, 1, p. 37-44

    Research output: Contribution to journalJournal articleResearchpeer-review

  27. Published

    Oral bioavailability and bone-sparing effects of estetrol in an osteoporosis model

    Coelingh Bennink, H. J. T., Heegaard, Anne-Marie, Visser, M., Holinka, C. F. & Christiansen, C., 2008, In: Climacteric. 11, 1, p. 2-14

    Research output: Contribution to journalJournal articleResearchpeer-review

  28. Published

    Palladium-catalyzed monoamination of dihalogenated benzenes

    Larsen, S. B., Bang-Andersen, B., Johansen, Tommy Nørskov & Jørgensen, M., 2008, In: Tetrahedron. 64, 13, p. 2938-2950

    Research output: Contribution to journalJournal articleResearchpeer-review

  29. Published

    Pegylated interferon alfa and ribavirin for 14 versus 24 weeks in patients with hepatitis C virus genotype 2 or 3 and rapid virological response

    Dalgard, O., Bjøro, K., Larsen, H. R., Bjornsson, E., Holberg-Petersen, M., Skovlund, E., Reichard, O., Myrvang, B., Sundelöf, B., Ritland, S., Hellum, K., Frydén, A., Florholmen, J. & Verbaan, H., 2008, In: Hepatology. 47, 1, p. 35-42

    Research output: Contribution to journalJournal articleResearchpeer-review

  30. Published

    Pharmacokinetic-Pharmacodynamic modeling of morphine and oxycodone concentrations and analgesic effect in a multimodal experimental pain model

    Staahl, C., Upton, R., Foster, D. J. R., Christrup, Lona Louring, Kristensen, K., Hansen, S. H., Arendt-Nielsen, L. & Drewes, A. M., 2008, In: Journal of Clinical Pharmacology. 48, 5, p. 619-631

    Research output: Contribution to journalJournal articleResearchpeer-review

  31. Published

    Pharmacokinetic-Pharmacodynamic relationships of cognitive and psychomotor effects of intravenous buprenorphine infusion in human volunteers

    Jensen, M. L., Sjøgren, P., Upton, R. N., Foster, D. J. R., Bonde, P., Graae, C., Skram, U., Stevner, L. L. S. & Christrup, Lona Louring, 2008, In: Basic & Clinical Pharmacology & Toxicology. 103, 1, p. 94-101

    Research output: Contribution to journalJournal articleResearchpeer-review

  32. Published

    Pharmacokinetics and pharmacodynamics of intranasal versus intravenous fentanyl in patients with pain after oral surgery

    Foster, D., Upton, R., Christrup, Lona Louring & Popper, L., 2008, In: Annals of Pharmacotherapy. 42, 10, p. 1380-1387

    Research output: Contribution to journalJournal articleResearchpeer-review

  33. Published

    Pharmacokinetics, efficacy, and tolerability of fentanyl following intranasal versus intravenous administration in adults undergoing third-molar extraction: A randomized, double-blind, double-dummy, two-way, crossover study

    Christrup, Lona Louring, Foster, D., Popper, L. D., Troen, T. & Upton, R., 2008, In: Clinical Therapeutics. 30, 3, p. 469-481

    Research output: Contribution to journalJournal articleResearchpeer-review

  34. Published

    Pharmacological characterization of ligands at recombinant NMDA receptor subtypes by electrophysiological recordings and intracellular calcium measurements

    Hansen, K. B., Bräuner, Hans & Egebjerg, J., 2008, In: Combinatorial Chemistry & High Throughput Screening. 11, 4, p. 304-315

    Research output: Contribution to journalJournal articleResearchpeer-review

  35. Published

    Pharmacological manipulation of extrasynaptic GABA transporters: implications for epilepsy management

    Madsen, K. K., Ebert, B., Larsson, O. M., Clausen, Rasmus Prætorius, Schousboe, Arne & White, H. S., 2008, In: Epilepsia. Suppl. 7, p. 347

    Research output: Contribution to journalConference abstract in journalResearch

  36. Published

    Phase transformation of erythromycin A dihydrate during fluid bed drying

    Römer, M., Heinämäki, J., Miroshnyk, I., Kivikero, N., Sandler, N., Rantanen, Jukka & Yliruusi, J., 2008, In: Journal of Pharmaceutical Sciences. 97, 9, p. 4020-4029

    Research output: Contribution to journalJournal articleResearchpeer-review

  37. Published

    Phylogenetic selection of Narcissus species for drug discovery

    Rønsted, Nina, Savolainen, V., Mølgaard, Per & Jäger, A. K., 2008, In: Biochemical Systematics and Ecology. 36, 5-6, p. 417-422

    Research output: Contribution to journalJournal articleResearchpeer-review

  38. Published

    Phylogeny, biogeography, and ecology of Ficus section Malvanthera (Moraceae)

    Rønsted, Nina, Weiblen, G. D., Savolainen, V. & Cook, J. M., 2008, In: Molecular Phylogenetics and Evolution. 48, 1, p. 12-22

    Research output: Contribution to journalJournal articleResearchpeer-review

  39. Published

    Phytochemical studies of plants used as antimalarials in Burkina Faso

    Traore, M., 2008, København: Det Farmaceutiske Fakultet. 160 p.

    Research output: Book/ReportPh.D. thesisResearch

  40. Published

    Poly(ethylene glycol)s generate complement activation products in human serum through increased alternative pathway turnover and a MASP-2-dependent process

    Hamad, I., Hunter, A. C., Szebeni, J. & Moghimi, S. M., 2008, In: Molecular Immunology. 46, 2, p. 225-232

    Research output: Contribution to journalJournal articleResearchpeer-review

  41. Published

    Polymeric nanocarriers for siRNA delivery: challenges and future prospects

    Cun, D., Jensen, L. B., Nielsen, Hanne Mørck, Moghimi, S. M. & Foged, Camilla, 2008, In: Journal of Biomedical Nanotechnology. 4, 3, p. 258-275

    Research output: Contribution to journalReviewResearch

  42. Published

    Positron emission tomography and its application to clinical oncology

    Honoré, P. G. H., 2008, In: European Journal of Oncology Pharmacy. 2, 2, p. 36-38

    Research output: Contribution to journalJournal articleResearchpeer-review

  43. Published

    Prediction of activation energies for aromatic oxidation by cytochrome P450

    Rydberg, P., Ryde, U. & Olsen, L., 2008, In: Journal of Physical Chemistry A. 112, 50, p. 13058-13065

    Research output: Contribution to journalJournal articleResearchpeer-review

  44. Published

    Prediction of the binding mode of biarylpropylsulfonamide allosteric AMPA receptor modulators based on docking, GRID molecular interaction fields and 3D-QSAR analysis

    Harpsøe, Kasper, Liljefors, T. & Balle, T., 2008, In: Journal of Molecular Graphics and Modelling. 26, 5, p. 874-883

    Research output: Contribution to journalJournal articleResearchpeer-review

  45. Published

    Prediction of the receptor conformation for iGluR2 agonist binding: QM/MM docking to an extensive conformational ensemble generated using normal mode analysis

    Sander, T., Liljefors, T. & Balle, T., 2008, In: Journal of Molecular Graphics and Modelling. 26, 8, p. 1259-1268

    Research output: Contribution to journalJournal articleResearchpeer-review

  46. Published

    Preface

    van de Weert, Marco & Møller, E. H., 2008, Immunogenicity of biopharmaceuticals. van de Weert, M. & Møller, E. H. (eds.). 1 ed. New York: Springer, p. v-vi

    Research output: Chapter in Book/Report/Conference proceedingPreface/postscriptResearch

  47. Published

    Probalistic ecological risk assessment of multiple pharmaceuticals in sewage treatment plant effluent

    Christensen, A. M., Baun, A. & Halling-Sørensen, B., 2008, World under stress: scientific and applied issues in environmental toxicology and chemistry. Society of Environmental Toxicology and Chemistry, p. 46-46

    Research output: Chapter in Book/Report/Conference proceedingConference abstract in proceedingsCommissioned

  48. Published

    Protein pharmaceuticals

    van de Weert, Marco & Møller, E. H., 2008, In: Drug Discovery Today: Technologies. 5, 2-3, p. 35-36

    Research output: Contribution to journalEditorialResearch

  49. Published

    Protein-protein interaktion: et nyt mål for udvikling af lægemidler

    Bach, Anders, Gottschalk, M., Kristensen, Anders Skov & Strømgaard, Kristian, 2008, In: Lægemiddelforskning. p. 10-12

    Research output: Contribution to journalJournal articleCommunication

  50. Published

    QSAR models for the human H+/peptide symporter, hPEPT1: Affinity prediction using alignment-independent descriptors

    Larsen, S. B., Jørgensen, Flemming Steen & Olsen, L., 2008, In: Journal of Chemical Information and Modeling. 48, 1, p. 233-241

    Research output: Contribution to journalJournal articleResearchpeer-review

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