Research areas

  1. Published

    Potentiating action of propofol at GABAA receptors of retinal bipolar cells

    Yue, L., Xie, A., Bruzik, K. S., Frølund, Bente, Qian, H. & Pepperberg, D. R., 1 Jan 2011, In: Investigative Ophthalmology & Visual Science. 52, 5, p. 2497-2509

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Purification, crystallization and preliminary X-ray diffraction of the G3BP1 NTF2-like domain

    Vognsen, T., Möller, I. R. & Kristensen, O., 1 Jan 2011, In: Acta Crystallographica. Section F: Structural Biology and Crystallization Communications Online. 67, Pt 1, p. 48-50

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Triazoloquinazolinediones as novel high affinity ligands for the benzodiazepine site of GABA(A) receptors

    Nilsson, J., Gidlöf, R., Nielsen, E. Ø., Liljefors, T., Nielsen, M. P. C. & Sterner, O., 1 Jan 2011, In: Bioorganic & Medicinal Chemistry. 19, 1, p. 111-121

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    The minor C-allele of rs2014355 in ACADS is associated with reduced insulin release following an oral glucose load

    Hornbak, M., Banasik, Karina, Justesen, Johanne Marie, Krarup, N. T., Sandholt, C. H., Andersson, Åsa, Sandbaek, A., Lauritzen, T., Pisinger, C., Witte, D. R., Sørensen, Thorkild I.A., Pedersen, Oluf Borbye & Hansen, Torben, 6 Jan 2011, In: BMC Medical Genetics. 12, 1, p. 4 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Intestinal drug delivery via hPEPT1 : in vitro and in silico evaluation of the realtionship between substrate, binding and translocation

    Omkvist, D. H., Feb 2011, Det Farmaceutiske Fakultet. 51 p.

    Research output: Book/ReportPh.D. thesisResearch

  6. Published

    Isolation of immunomodulatory triterpene acids from a standardized rose hip powder (Rosa canina L.)

    Saaby, Lasse, Jäger, A. K., Moesby, L., Hansen, E. W. & Christensen, Søren Brøgger, Feb 2011, In: Phytotherapy Research. 25, 2, p. 195-201

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Synthesis of new isoxazoline-based acidic amino acids and investigation of their affinity and selectivity profile at ionotropic glutamate receptors

    Pinto, A., Conti, P., Grazioso, G., Tamborini, L., Madsen, Ulf, Nielsen, Birgitte & De Micheli, C., 1 Feb 2011, In: European Journal of Medicinal Chemistry. 46, 2, p. 787-793

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Biophysical characterization of the complex between human papillomavirus E6 protein and synapse-associated protein 97

    Chi, C. N., Bach, Anders, Engström, Å., Strømgaard, Kristian, Lundström, P., Ferguson, N. & Jemth, P., 4 Feb 2011, In: Journal of Biological Chemistry. 286, 5, p. 3597-3606

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Expedient synthesis of 1,3-substituted benzene peptidomimetics

    Bach, Anders & Strømgaard, Kristian, 8 Feb 2011, In: Synthesis. 2011, 5, p. 807-815

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Flavonoids and the CNS

    Jäger, A. K. & Saaby, Lasse, 10 Feb 2011, In: Molecules. 16, 2, p. 1471-1485

    Research output: Contribution to journalReviewResearchpeer-review

  11. Published

    Functional and structural studies of neuronal D-serine transporter Asc1

    Wang, X., 10 Feb 2011, København: Det Farmaceutiske Fakultet. 148 p.

    Research output: Book/ReportPh.D. thesisResearch

  12. Published

    Medicinal chemistry of competitive kainate receptor antagonists

    Larsen, A. M. & Bunch, Lennart, 16 Feb 2011, In: ACS Chemical Neuroscience. 2, 2, p. 60-74

    Research output: Contribution to journalReviewResearchpeer-review

  13. Published

    Human phenotypically distinct TGFBI corneal dystrophies are linked to the stability of the fourth FAS1 domain of TGFBIp

    Runager, K., Basaiawmoit, R. V., Deva, T., Andreasen, M., Valnickova, Z., Sørensen, C. S., Karring, H., Thøgersen, I. B., Christiansen, G., Underhaug, J., Kristensen, T., Nielsen, N. C., Klintworth, G. K., Otzen, D. E. & Enghild, J. J., 18 Feb 2011, In: The Journal of Biological Chemistry. 286, 7, p. 4951-4958

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. Published

    G protein- and agonist-bound serotonin 5-HT2A receptor model activated by steered molecular dynamics simulations

    Ísberg, V., Balle, T., Sander, T., Jørgensen, Flemming Steen & Gloriam, David E., 28 Feb 2011, In: Journal of Chemical Information and Modeling. 51, 2, p. 315-325

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    European new safe and innovative medicines initiatives: history and progress (through December 2009)

    Bjerrum, Ole Jannik & H. Linden, H., Mar 2011, Translational medicine and drug discovery. Cambridge: Cambridge University Press, p. 265-288 23 p.

    Research output: Chapter in Book/Report/Conference proceedingBook chapterCommunication

  16. Published

    Metabolic profiling of Rhodiola rosea rhizomes by 1H NMR spectroscopy

    Ioset, K. N., Nyberg, N. T., Van Diermen, D., Malnoe, P., Hostettmann, K., Shikov, A. N. & Jaroszewski, J. W., Mar 2011, In: Phytochemical Analysis. 22, 2, p. 158-165

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    Cell-permeable and plasma-stable peptidomimetic inhibitors of the postsynaptic density-95/N-methyl-D-aspartate receptor interaction

    Bach, Anders, Eildal, J. N. N., Stuhr-Hansen, N., Deeskamp, R., Gottschalk, M., Pedersen, S. W., Kristensen, Anders Skov & Strømgaard, Kristian, 10 Mar 2011, In: Journal of Medicinal Chemistry. 54, 5, p. 1333-1346

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    Amaryllidaceae alkaloids from the Australasian tribe Calostemmateae with acetylcholinesterase inhibitory activity

    Søvsø Jensen, B., Christensen, Søren Brøgger, Jäger, A. K. & Rønsted, Nina, Apr 2011, In: Biochemical Systematics and Ecology. 39, 2, p. 153-155

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    Glutamate receptor agonists: stereochemical aspects

    Vogensen, S. B., Greenwood, J. R., Bunch, Lennart & Clausen, Rasmus Prætorius, Apr 2011, In: Current Topics in Medicinal Chemistry. 11, 7, p. 887-906

    Research output: Contribution to journalReviewResearchpeer-review

  20. Published

    Discovery of benzamide analogues as a novel class of 5-HT3 receptor agonists

    Jørgensen, Charlotte Grube, Frølund, Bente, Kehler, J. & Jensen, Anders A., 4 Apr 2011, In: ChemMedChem. 6, 4, p. 725-736

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    ZP2307, a novel cyclic PTH(1-17) analog, reversed established osteopenia in adult ovariectomized rats

    Vääräniemi, J., Morko, J., Peng, Z., Rissanen, J. P., Suominen, M. I., Fagerlund, K. M., Suutari, T. A., Boonen, H. C. M., Neerup, T. S., Bak, H. H. & Halleen, J. M., 7 Apr 2011. 1 p.

    Research output: Contribution to conferencePosterResearch

  22. Published

    Electrophilic organic selenium reagents: protonated seleninic acids as precursors for unsymmetrical aromatic selenides

    Stuhr-Hansen, N., Sølling, Theis Ivan & Henriksen, L., 8 Apr 2011, In: Tetrahedron. 67, 14, p. 2633-2643

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    Pharmacological properties of Anagallis arvensis L. ("scarlet pimpernel") and Anagallis foemina Mill. ("blue pimpernel") traditionally used as wound healing remedies in Navarra (Spain)

    López, V., Jäger, A. K., Akerreta, S., Cavero, R. Y. & Calvo, M. I., 12 Apr 2011, In: Journal of Ethnopharmacology. 134, 3, p. 1014-1017

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Comparative pharmacokinetics between a microdose and therapeutic dose for clarithromycin, sumatriptan, propafenone, paracetamol (acetaminophen) and phenobarbital in human volunteers

    Lappin, G., Shishikura, Y., Jochemsen, R., Weaver, R. J., Gesson, C., Houston, J. B., Oosterhuis, B., Bjerrum, Ole Jannik, Grynkiewicz, G., Alder, J., Rowland, M. & Garner, C., 20 Apr 2011, In: European Journal of Pharmaceutical Sciences. 43, 3, p. 141-150 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    1,2,3-triazoles in peptidomimetic chemistry

    Pedersen, D. S. & Abell, A., May 2011, In: European Journal of Organic Chemistry. 2011, 13, p. 2399-2411

    Research output: Contribution to journalReviewResearchpeer-review