Research areas

  1. Published

    Scientific social responsibility: a call to arms

    Krogsgaard-Larsen, Povl, Thostrup, P. & Besenbacher, F., 11 Nov 2011, In: Angewandte Chemie International Edition. 50, 46, p. 10738-10740

    Research output: Contribution to journalComment/debateResearch

  2. Published

    Amino triazolo diazepines (Ata) as constrained histidine mimics

    Buysse, K., Farard, J., Nikolaou, A., Vanderheyden, P., Vauquelin, G., Pedersen, D. S., Tourwé, D. & Ballet, S., 16 Nov 2011, In: Organic Letters. 13, 24, p. 6468-6471

    Research output: Contribution to journalLetterResearchpeer-review

  3. Published

    Chemogenomic discovery of allosteric antagonists at the GPRC6A receptor

    Gloriam, David E., Wellendorph, Petrine, Johansen, L. D., Thomsen, A. R. B., Phonekeo, K., Pedersen, D. S. & Bräuner, Hans, 23 Nov 2011, In: Chemistry & Biology. 18, 11, p. 1489-1498

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Small molecules from spiders used as chemical probes

    Olsen, C. A., Kristensen, Anders Skov & Strømgaard, Kristian, 25 Nov 2011, In: Angewandte Chemie International Edition. 50, 48, p. 11296-11311

    Research output: Contribution to journalReviewResearchpeer-review

  5. Published

    From retrospective assessment to prospective decisions in natural product isolation: HPLC-SPE-NMR analysis of Carthamus oxyacantha

    Kongstad, Kenneth Thermann, Wubshet, S. G., Nyberg, N. T. & Jaroszewski, J. W., 28 Nov 2011, In: Journal of Natural Products. 74, 11, p. 2454-2461

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    An in vitro assay based on surface plasmon resonance to predict the in vivo circulation kinetics of liposomes

    Crielaard, B. J., Yousefi, A., Schillemans, J. P., Vermehren, C., Buyens, K., Braeckmans, K., Lammers, T. & Storm, G., Dec 2011, In: Journal of Controlled Release. 156, 3, p. 307-314

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published
  8. Published

    Computeren forudsiger lægemidlers omdannelse i leveren

    Rydberg, P. & Olsen, L., Dec 2011, In: Lægemiddelforskning. 2011, p. 44-46

    Research output: Contribution to journalJournal articleCommunication

  9. Published

    Funktionelle fibriller som depotmedicin mod prostatakræft

    Jensen, M. G., van Maarschalkerweerd, A. & Gottschalk, T., Dec 2011, In: Lægemiddelforskning. 2011, p. 20-22

    Research output: Contribution to journalJournal articleCommunication

  10. Published

    Gendannelse af ødelagt væv med stamceller

    Møller, E. H., Wen, Y. & Nielsen, Hanne Mørck, Dec 2011, In: Lægemiddelforskning. 2011, p. 13-15

    Research output: Contribution to journalJournal articleCommunication

  11. Published

    Genetisk nanomedicin til behandling af leddegigt

    Foged, Camilla, Jensen, L. B. & Nielsen, Hanne Mørck, Dec 2011, In: Lægemiddelforskning. p. 7-9

    Research output: Contribution to journalJournal articleCommunication

  12. Published

    Massespektrometri viser fordelingen af lægemiddelstoffer i planter og væv

    Janfelt, Christian, Thunig, J., Li, B., Andersen, N. W., Hansen, Harald S. & Hansen, S. H., Dec 2011, In: Lægemiddelforskning. 2011, p. 10-12

    Research output: Contribution to journalJournal articleCommunication

  13. Published

    Medicinalplanter og abort: ny viden kan hjælpe afrikanske kvinder

    Jäger, A., Kristiansen, Uffe & Rasch, V., Dec 2011, In: Lægemiddelforskning. 2011, p. 23-25

    Research output: Contribution to journalJournal articleCommunication

  14. Published

    Målrettet fisketur i hjernen giver ny viden om Fantasys virkningssted

    Villumsen, I. S., Vogensen, S. B., Frølund, Bente, Clausen, Rasmus Prætorius & Wellendorph, Petrine, Dec 2011, In: Lægemiddelforskning. 2011, p. 26-28

    Research output: Contribution to journalJournal articleCommunication

  15. Published

    Nanobodies fra kameler - En ny klasse antistoffer til diagnostik og behandling

    Skottrup, P. D., Clausen, Rasmus Prætorius & Riise, E., Dec 2011, In: Lægemiddelforskning. 2011, p. 4-6

    Research output: Contribution to journalJournal articleCommunication

  16. Published

    A pinch of sodium

    Müller, M. S., 1 Dec 2011, In: Nature Chemistry. 3, 12, p. 974

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    Neuron-glia interactions in glutamatergic neurotransmission: roles of oxidative and glycolytic adenosine triphosphate as energy source

    Schousboe, Arne, Sickmann, H. M., Bak, Lasse Kristoffer, Schousboe, I., Jajo, F. S., Faek, S. A. A. & Waagepetersen, Helle S., 1 Dec 2011, In: Journal of Neuroscience Research. 89, 12, p. 1926-34 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    Synthesis of the thiazole-thiazoline fragment of largazole analogues

    Diness, Frederik, Nielsen, D. S. & Fairlie, D. P., 2 Dec 2011, In: Journal of Organic Chemistry. 76, 23, p. 9845-9851

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    Characterization of upper thoracic spinal neurons receiving noxious cardiac and/or somatic inputs in diabetic rats

    Ghorbani, M. L. M., Qin, C., Wu, M., Farber, J. P., Sheykhzade, Majid, Fjalland, B., Nyborg, N. C. B. & Foreman, R. D., 7 Dec 2011, In: Autonomic Neuroscience: Basic and Clinical. 165, 2, p. 168-177

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    3-Hydroxy-2'-methoxy-6-methylflavone: a potent anxiolytic with a unique selectivity profile at GABA(A) receptor subtypes

    Karim, N., Gavande, N., Wellendorph, Petrine, Johnston, G. A. R., Hanrahan, J. R. & Chebib, M., 15 Dec 2011, In: Biochemical Pharmacology. 82, 12, p. 1971-1983

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    New cholesterol esterase inhibitors based on rhodanine and thiazolidinedione scaffolds

    Heng, S., Tieu, W., Hautmann, S., Kuan, K., Pedersen, D. S., Pietsch, M., Gütschow, M. & Abell, A. D., 15 Dec 2011, In: Bioorganic & Medicinal Chemistry. 19, 24, p. 7453-7463

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Acetylcholine binding protein as model of alpha4beta2 nicotinic acetylcholine receptors: Structural and functional characterization

    Rohde, L. A. H., 19 Dec 2011, København: Det Farmaceutiske Fakultet. 104 p.

    Research output: Book/ReportPh.D. thesisResearch

  23. Published

    In vitro efficacy testing of praziquantel, ivermectin, and oxfendazole against Taenia Solium cysts

    Cederberg, S., Sikasunge, C. S., Andersson, Åsa & Johansen, M. V., 2012, In: Journal of Parasitology Research. 2012, 4 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    In vitro release from oil injectabels for intra-articular administration: importance of interfacial area, diffusivity and partitioning

    Thing, M. A., Larsen, C. S., Østergaard, Jesper, Jensen, H. & Larsen, Susan Weng, 2012, In: European Journal of Pharmaceutical Sciences. 45, 3, p. 351-357

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    A 3D-QSAR-driven approach to binding mode and affinity prediction

    Tosco, P. & Balle, T., 2012, In: Journal of Chemical Information and Modeling. 52, 2, p. 302-307

    Research output: Contribution to journalJournal articleResearchpeer-review

  26. Published

    A robust force field based method for calculating conformational energies of charged drug-like molecules

    Pøhlsgaard, J., Harpsøe, Kasper, Jørgensen, Flemming Steen & Olsen, L., 2012, In: Journal of Chemical Information and Modeling. 52, 2, p. 409-419

    Research output: Contribution to journalJournal articleResearchpeer-review

  27. Published

    Absorption difference between diacylglycerol oil and butter blend containing deacylglycerol oil

    Kristensen, J. B., Jørgensen, H. & Mu, Huiling, 2012, In: European Journal of Lipid Science and Technology. 114, 2, p. 146-152

    Research output: Contribution to journalJournal articleResearchpeer-review

  28. Published

    An electrochemical approach to protein adsorption at charged interfaces

    Hartvig, R. A., 2012, København: Det Farmaceutiske Fakultet. 127 p.

    Research output: Book/ReportPh.D. thesisResearch

  29. Published

    Assessing element-specific patterns of bioaccumulation across New England lakes

    Ward, D. M., Mayes, B., Stürup, Stefan, Folt, C. L. & Chen, C. Y., 2012, In: Science of the Total Environment. 421-422, 3-4, p. 230-237

    Research output: Contribution to journalJournal articleResearchpeer-review

  30. Published

    Behaviour of HPMC compacts investigated using UV-imaging

    Pekka Pajander, J., Baldursdottir, S. G., Rantanen, Jukka & Østergaard, Jesper, 2012, In: International Journal of Pharmaceutics. 427, 2, p. 345-353

    Research output: Contribution to journalJournal articleResearchpeer-review

  31. Published

    Characterization of bupivacaine-loaded formulations based on liquid crystalline phases and microemulsions: the effect of lipid composition

    Yaghmur, Anan, Rappolt, M., Østergaard, Jesper, Larsen, C. S. & Larsen, Susan Weng, 2012, In: Langmuir. 28, 5, p. 2881-2889

    Research output: Contribution to journalJournal articleResearchpeer-review

  32. Published

    Comparison of polymeric siRNA nanocarriers in murine LPS-activated macrophage cell line: Gene silencing, toxicity and off-target gene expression

    Jensen, L. B., Griger, J., Naeye, B., Varkouhi, A. K., Raemdonck, K., Schiffelers, R., Lammers, T., Storm, G., Smedt, S. C. D., Sproat, B. S., Nielsen, Hanne Mørck & Foged, Camilla, 2012, In: Pharmaceutical Research. 29, p. 669-682

    Research output: Contribution to journalJournal articleResearchpeer-review

  33. Published

    Correlation between enzyme activity an stability of a protease, an alpha-amaylase and a lipase in a simplified liquid laundry detergent system, determined by differential scanning calorimetry

    Lund, H., Kaasgaard, S. G., Skagerlind, P., Jørgensen, Lene, Jørgensen, C. I. & van de Weert, Marco, 2012, In: Journal of Surfactants and Detergents. 15, p. 9-21

    Research output: Contribution to journalJournal articleResearchpeer-review

  34. Published

    Delivery of dermatan sulfate from polyelectrolyte complex-containing alginate composite microspheres for tissue regeneration

    Wen, Y., Grøndahl, L., Gallego, M. R., Jørgensen, Lene, Møller, E. H. & Nielsen, Hanne Mørck, 2012, In: Biomacromolecules. 13, p. 905-917

    Research output: Contribution to journalJournal articleResearchpeer-review

  35. Published

    Design of an inhalable dry powder formulation of DOTAP-modified PLGA nanoparticles loaded with siRNA

    Jensen, D. M. K., Jensen, L. B., Koocheki, S., Cun, D., Nielsen, Hanne Mørck, Foged, Camilla & Bengtson, L., 2012, In: Journal of Controlled Release. 157, 1, p. 141-148

    Research output: Contribution to journalJournal articleResearchpeer-review

  36. Published

    Design of cyclic RKKH peptide-conjugated PEG liposomes targeting the integrin a2ß1 receptor

    Knudsen, N. Ø., Schiffelers, R. M., Jørgensen, Lene, Hansen, J., Frøkjær, Sven & Foged, Camilla, 2012, In: International Journal of Pharmaceutics. 428, 1-2, p. 171-177

    Research output: Contribution to journalJournal articleResearchpeer-review

  37. Published

    Design space approach in the optimization of the spray-drying process

    Lebrun, P., Krier, F., Mantanus, J., Grohganz, Holger, Yang, Mingshi, Rozet, E., Boulanger, B., Evrard, B., Rantanen, Jukka & Hubert, P., 2012, In: European Journal of Pharmaceutics and Biopharmaceutics. 80, 1

    Research output: Contribution to journalJournal articleResearchpeer-review

  38. Published

    Drugs for the neglected disease malaria based on natural products

    Christensen, Søren Brøgger & Bygbjerg, Ib Christian, 2012, Bioactive compounds from natural sources: natural products as lead compounds in drug discovery. Tringali, C. (ed.). 2 ed. Boca Raton: CRC Press, p. 525-550

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  39. Published

    Estimating intestinal absorption of inorganic selenium compounds by in vitro flux and biotransformation studies in Caco-2 cells and ICP-MS detection

    Gammelgaard, Bente, Rasmussen, L. H., Gabel-Jensen, C. & Steffansen, B., 2012, In: Biological Trace Element Research. 145, 2, p. 248-256

    Research output: Contribution to journalJournal articleResearchpeer-review

  40. Published

    Fast, selective, and sensitive analysis of low-abundance peptides in human plasma by electromembrane exctraction

    Balchen, M., Lund, H., Reubsaet, L. & Pedersen-Bjergaard, Stig, 2012, In: Analytica Chimica Acta. 716, p. 16-23

    Research output: Contribution to journalJournal articleResearchpeer-review

  41. Published

    Forced degradation of therapeutic proteins

    Hawe, A., Wiggenhorn, M., van de Weert, Marco, Garbe, J. H. O., Mahler, H. & Jiskoot, W., 2012, In: Journal of Pharmaceutical Sciences. 101, 3, p. 895-913

    Research output: Contribution to journalReviewResearchpeer-review

  42. Published

    Formation of dielectric layers and charge regulation in protein adsorption at biomimetic interfaces

    Hartvig, R. A., van de Weert, Marco, Østergaard, Jesper, Jørgensen, Lene & Jensen, H., 2012, In: Langmuir. 28, 3, p. 1804-1815

    Research output: Contribution to journalJournal articleResearchpeer-review

  43. Published

    How to engage experienced medicine users at the counter for a pharmacy-based asthma inhaler service

    Kaae, Susanne & Nørgaard, Lotte Stig, 2012, In: International Journal of Pharmacy Practice. 20, p. 99-106

    Research output: Contribution to journalJournal articleResearchpeer-review

  44. Published

    Human urinary excretion and metabolism of 82Se-enriched selenite and selenate determined by LC-ICP-MS

    Gammelgaard, Bente, Stürup, Stefan & Christensen, M. V., 2012, In: Metallomics. 4, 2, p. 149-155

    Research output: Contribution to journalJournal articleResearchpeer-review

  45. Published

    Håb om at ramme latente bakterier i deres skjul

    Bahnsen, J. S., Water, J. J., Foged, Camilla, Franzyk, Henrik & Nielsen, Hanne Mørck, 2012, In: Lægemiddelforskning 2012. 2012, p. 12-14

    Research output: Contribution to journalJournal articleResearch

  46. Published

    In vitro digestion testing of lipid-based delivery systems: calcium ions combine with fatty acids liberated from triglyceride rich lipid solutions to form soaps and reduce the solubilization capacity of colloidal digestion products

    Devraj, R., Williams, H. D., Warren, D. B., Mullertz, Anette , Porter, C. J. H. & Pouton, C. W., 2012, In: International Journal of Pharmaceutics. 441, 1-2, p. 323-333

    Research output: Contribution to journalJournal articleResearchpeer-review

  47. Published

    Influence of lipid composition and drug load on the in vitro performance of self-nanoemulsifying drug delivery systems

    Thomas, N., Mullertz, Anette , Graf, A. & Rades, T., 2012, In: Journal of Pharmaceutical Sciences. 101, 5, p. 1721-1731

    Research output: Contribution to journalJournal articleResearchpeer-review

  48. Published

    Insights into intermediate phases of human intestinal fluids visualized by atomic force microscopy and cryo-transmission electron microscopy ex vivo

    Mullertz, Anette , Fatouros, D. G., Smith, J. R., Vertzoni, M. & Reppas, C., 2012, In: Molecular Pharmaceutics. 9, 2, p. 237-247

    Research output: Contribution to journalJournal articleResearchpeer-review

  49. Published

    Interaction of peptidomimetics with bilayer membranes: biophysical characterization and cellular uptake

    Jing, X., Kasimova, M. R., Simonsen, A. H., Jørgensen, Lene, Malmsten, M., Franzyk, Henrik & Foged, Camilla, 2012, In: Langmuir. 28, 11, p. 5167-5175

    Research output: Contribution to journalJournal articleResearchpeer-review

  50. Published

    Internal correction of spectral interferences and mass bias for selenium metabolism studies using enriched stabel isotopes in combination with multiple linear regression

    Lunøe, K., Martinez-Sierra, J. G., Gammelgaard, Bente & Alonso, J. I. G., 2012, In: Analytical and Bioanalytical Chemistry. 402, 9, p. 2749-2763

    Research output: Contribution to journalJournal articleResearchpeer-review